[J60384] CAS 65391-42-6 | Bestatin hydrochloride, 98% | Alfa
0 ₩
Brand: Alfa Aesar
65391-42-6 | C16H25ClN2O4 | hydrogen (2R,4S,5R)-2,5-diamino-4-hydroxy-2-(2-methylpropyl)-3-oxo-6-phenylhexanoic acid chloride
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Chemical Identifiers
CAS
65391-42-6
Molecular Weight (g/mol)
344.84
Synonym
hydrogen (2R,4S,5R)-2,5-diamino-4-hydroxy-2-(2-methylpropyl)-3-oxo-6-phenylhexanoic acid chloride
SMILES
[H+].[Cl-].CC(C)C[C@](N)(C(O)=O)C(=O)[C@@H](O)[C@H](N)CC1=CC=CC=C1
InChI Key
JQOATSUOLWQWKR-KHUBKBNHSA-N
Molecular Formula
C16H25ClN2O4
IUPAC Name
hydrogen (2R,4S,5R)-2,5-diamino-4-hydroxy-2-(2-methylpropyl)-3-oxo-6-phenylhexanoic acid chloride
Specifications
Assay from Suppliers CofA
≥97.5%
Form
Powder
설명
Bestatin is an inhibitor of amino peptidases and a potent, irreversible inhibitor of LTA4 hydrolase. It inhibits the amino peptidase activity of LTA4 hydrolase with a Ki value of 201 nM. It offers promise as a novel analgesic because it protects endogenous opioid peptides against degradation. It does not inhibit carboxypeptidases.
This Thermo Scientific Chemicals brand product was originally part of the Alfa Aesar product portfolio. Some documentation and label information may refer to the legacy brand. The original Alfa Aesar product / item code or SKU reference has not changed as a part of the brand transition to Thermo Scientific Chemicals.
Applications
Bestatin is an inhibitor of amino peptidases and a potent, irreversible inhibitor of LTA4 hydrolase. It inhibits the amino peptidase activity of LTA4 hydrolase with a Ki value of 201 nM. It offers promise as a novel analgesic because it protects endogenous opioid peptides against degradation. It does not inhibit carboxypeptidases.
Bestatin is an inhibitor of amino peptidases and a potent, irreversible inhibitor of LTA4 hydrolase. It inhibits the amino peptidase activity of LTA4 hydrolase with a Ki value of 201 nM. It offers promise as a novel analgesic because it protects endogenous opioid peptides against degradation. It does not inhibit carboxypeptidases.
Solubility
Soluble in water (4 mg/ml, warm), DMSO (>25 mg/ml), methanol, acetic acid, dimethyl formamide, and 100% ethanol.
Notes
Store in cool, dry place in a tightly sealed container. Store away from oxidizing agents.
Other References:
Beilstein:4628066
GHS Hazard and Precautionary Statements
Hazard Statements:
Risk & Safety
TSCA:No
경고:RUO – Research Use Only
CAS65391-42-6FORMULAC16H25ClN2O4MDLMFCD00058004
| Pakage | 25mg, 5mg |
|---|---|
| brand | Alfa Aesar |
